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Fragment-Hopping-Based Discovery of a Novel Chemical Series of Proto-Oncogene PIM-1 Kinase Inhibitors
ArticleAbstract: A new chemical series, triazolo[4,5-b]pyridines, has been identified as an inhibitor of PIM-1 by a cPalabras claves:Autores:Albarran M.I., Alvarez R.M., Antonio Salgado, Bischoff J.R., Blanco C., Kurz G., Ortega M.A., Oyarzabal J., Pastor J., Pevarello P., Rabal O., Saluste G.Fuentes:scopusExome sequencing of plasma DNA portrays the mutation landscape of colorectal cancer and discovers mutated VEGFR2 receptors as modulators of antiangiogenic therapies
ArticleAbstract: Purpose: Despite the wide use of antiangiogenic drugs in the clinical setting, pbkp_redictive biomarPalabras claves:Autores:Albarran M.I., Alvarez R., Banos N., Blanco-Aparicio C., Camacho-Artacho M., Cubillo A., De Martino A., Domínguez O., Durán Y., Garralda E., Hidalgo M., Lietha D., Martínez-Torrecuadrada J.L., Mitsi M., Monsech J., Otero A., Perea S., Pons T., Sanchez-Perez T., Sarno F., Toledo R.A., Vega E., Victoria Maritza Cevallos BonillaFuentes:scopus