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Colchicine for the primary prevention of cardiovascular events
ReviewAbstract: Objectives: This is a protocol for a Cochrane Review (intervention). The objectives are as follows:.Palabras claves:Autores:Alegría E., Correa-Pérez A., de Sanctis J.B., Martí-Amarista C.E., Monge Martín D., Prof. Arturo Martí Carvajal MD MSc Ph.D iD, Ricardo Hidalgo-Ottolenghi, Riera Lizardo R.J.Fuentes:googlescopusCytotoxic activity of seco-entkaurenes from Croton caracasana on human cancer cell lines
ArticleAbstract: In the course of searching for bioactive compounds from Croton species from Venezuela, two seco-entkPalabras claves:Croton caracasana, Cytotoxic, euphorbiaceae, seco-entkaurenesAutores:Alírica Isabel Suárez, Arvelo F.A., Chavez K., Compagnone R.S., de Sanctis J.B., Mateu E., Mijares M.R., Muñoz A., Sojo F.J.Fuentes:scopusNovel 7-Chloro-(4-thioalkylquinoline) Derivatives: Synthesis and Antiproliferative Activity through Inducing Apoptosis and DNA/RNA Damage
ArticleAbstract: A series of 78 synthetic 7-chloro-(4-thioalkylquinoline) derivatives were investigated for cytotoxicPalabras claves:antiproliferative activity, cell cycle, DNA/RNA damage, Sulfanyl-Sulfinyl-Sulfonyl groups, synthesis of 4-thioalkylquinolineAutores:Bruno-Colmenarez J., Charris J.E., de Sanctis J.B., Deffieux D., Džubák P., Esteban Fernández-Moreira, Gurská S., Gutiérrez J.E., Hajdůch M., Hegira Ramírez, Mijares M.R., Pouységu L., Quideau S., Rodríguez M.A., Rojas L.B.Fuentes:scopusPharmacological properties of thalidomide and its analogues
ArticleAbstract: Thalidomide and its immunomodulatory imide drugs (IMiDs) analogues CC-5013 (Revlimid™, Lenalidomide)Palabras claves:Actimid, Angiogenesis, cytokines, DIABÉTES, Imids, Lenalidomide, Multiple myeloma, Pomalidomide, Prostate cancer, Revlimid, ThalidomideAutores:Alírica Isabel Suárez, Compagnone R.S., de Sanctis J.B., Garmendia J., Mijares M.R., Moreno D., Salazar-Bookaman M.Fuentes:scopusSpecialized pro-resolving lipid mediators: The future of chronic pain therapy?
ReviewAbstract: Chronic pain (CP) is a severe clinical entity with devastating physical and emotional con-sequencesPalabras claves:Central nervous system sensitization, Chronic pain, Eicosanoids, inflammation, Long-term poten-tiation, Nociception, Omega 3 fatty acids, pain management, Polyunsaturated fatty acids, Specialized pro-resolving lipid mediatorsAutores:Chávez-Castillo M., de Sanctis J.B., Durán P., Garrido B., Manzano A., Ortega A., Rojas M., Rojas-Gómez D.M., Salazar-Vílchez J., Silva A., Torres L.C., Valmore BermúdezFuentes:scopusSynthesis and antimalarial and anticancer evaluation of 7-chlorquinoline-4-thiazoleacetic derivatives containing aryl hydrazide moieties
ArticleAbstract: Twelve 7-chloroquinoline derivatives were designed and synthesized using the principle of molecularPalabras claves:Antimalarial, Antiproliferative, apoptosis, hydrazides, quinoline, thiazolAutores:Celis C., Charris J.E., de Sanctis J.B., Esteban Fernandez, Hegira Ramírez, Martinez G.P., Mayora S., Mijares M.R., Rodrigues J.R.Fuentes:scopusSynthesis and biological activity of 2-[2-(7-chloroquinolin-4-ylthio)-4-methylthiazol-5-yl]-N-phenylacetamide derivatives as antimalarial and cytotoxic agents
ArticleAbstract: A novel series of 2-[2-(7-chloroquinolin-4-ylthio)-4-methylthiazol-5-yl]-N-phenylacetamide derivativPalabras claves:ANTICANCER, Antimalarial, plasmodium, quinoline, thiazoleacetic acidAutores:Charris J.E., de Sanctis J.B., Hegira Ramírez, Mijares M.R., Rodrigues J.R.Fuentes:scopusSynthesis, Leishmanicidal, Trypanocidal, Antiproliferative Assay and Apoptotic Induction of (2-Phenoxypyridin-3-yl)naphthalene-1(2H)-one Derivatives
ArticleAbstract: The coexistence of leishmaniasis, Chagas disease, and neoplasia in endemic areas has been extensivelPalabras claves:apoptosis, Cáncer, chalcone, leishmaniasis, TRYPANOSOMA CRUZIAutores:Ángel J.E., Blanco Z., Celis C., Charris J.E., de Sanctis J.B., Džubák P., Esteban Fernández-Moreira, García Y., Gurská S., Hajdůch M., Hegira Ramírez, Jhonny Correa-Abril, Martinez G.P., Mijares M.R., Mijoba A., Nahum Herrera, Serrano X., Yonathan De J. ParraFuentes:scopus