Mostrando 4 resultados de: 4
Filtros aplicados
Subtipo de publicación
Article(4)
Publisher
Journal of Medicinal Chemistry(2)
Amino Acids(1)
Bioorganic and Medicinal Chemistry Letters(1)
Origen
scopus(4)
A BODIPY-embedding miltefosine analog linked to cell-penetrating Tat(48-60) peptide favors intracellular delivery and visualization of the antiparasitic drug
ArticleAbstract: Therapeutic application of many drugs is often hampered by poor or denied access to intracellular taPalabras claves:BODIPY, cell-penetrating peptide, Dual fluorescent labeling, Miltefosine, Monitoring of intracellular drug delivery, Reversion of resistanceAutores:Abengózar M.Á., Amat-Guerri F., Andreu D., B. G. De la Torre, Hornillos V., Luque-Ortega J.R., Rivas L., Ulises Acuña A.Fuentes:scopusSequence inversion and phenylalanine surrogates at the β-Turn enhance the antibiotic activity of gramicidin S
ArticleAbstract: A series of gramicidin S (GS) analogues have been synthesized where the Phe (i + 1) and Pro (i + 2)Palabras claves:Autores:Andreu D., B. G. De la Torre, Cativiela C., Fernández-Reyes M., Jiménez A.I., Jiménez M.A., Rivas L., Santiveri C.M., Solanas C.Fuentes:scopusSynthesis of 16-mercaptohexadecylphosphocholine, a miltefosine analog with leishmanicidal activity
ArticleAbstract: The alkylphosphocholine miltefosine (n-hexadecylphosphocholine, MT) has been introduced recently asPalabras claves:Hexadecylphosphocholine, LEISHMANIA, Mercaptophosphocholine, Miltefosine, ParasiticideAutores:Acuña A.U., Amat-Guerri F., Andreu D., B. G. De la Torre, Hornillos V., Rivas L., Saugar J.M.Fuentes:scopusTherapeutic index of gramicidin S is strongly modulated by D-phenylalanine analogues at the β-turn
ArticleAbstract: Analogues of the cationic antimicrobial peptide gramicidin S (GS), cyclo(Val-Orn-Leu-D-Phe-Pro)2, wiPalabras claves:Autores:Andreu D., B. G. De la Torre, Cativiela C., Fernández-Reyes M., Jiménez A.I., Jiménez M.A., Rivas L., Santiveri C.M., Solanas C.Fuentes:scopus