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Design and Synthesis of Broad Spectrum Trypanosomatid Selective Inhibitors
ArticleAbstract: Neglected tropical diseases caused by parasitic infections are an ongoing and increasing concern thaPalabras claves:chemical tools, drug design, Natural products, photoaffinity, TrypanosomatidAutores:Florence G.J., Fraser A.L., Gould E.R., King E.F.B., Smith T.K., Stefanie K. Menzies, Tulloch L.B., Zacharova M.K.Fuentes:scopusDirect and indirect approaches to identify drug modes of action
ReviewAbstract: Phenotypic assays are becoming increasingly more common among drug discovery practices, expanding drPalabras claves:affinity chromatography, drug mode of action, Genomics, Metabolomics, photo-affinity labeling, proteomics, target ID, transcriptomicsAutores:Coron R.P., Florence G.J., Roberts M.D., Smith T.K., Stefanie K. Menzies, Tulloch L.B.Fuentes:scopusThe trypanosome alternative oxidase: A potential drug target?
ReviewAbstract: New drugs against Trypanosoma brucei, the causative agent of Human African Trypanosomiasis, are urgePalabras claves:chemotherapy, Drug Discovery, human African trypanosomiasis, Sleeping sickness, Trypanosoma brucei, Trypanosome alternative oxidaseAutores:Florence G.J., Smith T.K., Stefanie K. Menzies, Tulloch L.B.Fuentes:scopus