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Current tendencies in antimicrobial research: Medicinal chemistry of antibacterial agents and advances in the use of computational methodologies
OtherAbstract:Palabras claves:Autores:Alejandro Speck-Planche, Natalia Dias Soeiro Cordeiro M., Scotti M.T.Fuentes:scopusMulti-target Drug Discovery via PTML Modeling: Applications to the Design of Virtual Dual Inhibitors of CDK4 and HER2
ArticleAbstract: Background: Cyclin-dependent kinase 4 (CDK4) and the human epidermal growth factor receptor 2 (HER2)Palabras claves:Artificial Neural Network, Cáncer, Fragment, Local contributions, Pseudo-linear equation, PTML model, virtual designAutores:Alejandro Speck-Planche, Kleandrova V.V., Scotti L., Scotti M.T.Fuentes:scopusNosocomial infections: An increasing challenge to medicinal chemistry
OtherAbstract:Palabras claves:Autores:Alejandro Speck-Planche, Natalia Dias Soeiro Cordeiro M., Scotti M.T.Fuentes:scopusIn silico studies for bacterystic evaluation against staphylococcus aureus of 2-naphthoic acid analogues
ArticleAbstract: Background: Staphylococcus aureus is a gram-positive spherical bacterium commonly present in nasal fPalabras claves:2-Naphthoic Acid Analogues, Cytotoxicity risks, KNIME Analytics Platform, Lipinski rule, PHENOLIC COMPOUNDS, STAPHYLOCOCCUS AUREUSAutores:Alejandro Speck-Planche, Costa Barros R.P., Messias Monteiro A.F., Scotti L., Scotti M.T.Fuentes:scopusIndirect-Acting Pan-Antivirals vs. Respiratory Viruses: A Fresh Perspective on Computational Multi-Target Drug Discovery
ArticleAbstract: Respiratory viruses continue to afflict mankind. Among them, pathogens such as coronaviruses [includPalabras claves:antiviral, Caspase-1, Coronaviruses, Indirect-acting pan-antiviral, influenza, multi-target, PTML, Sting, TLR7, TNF-αAutores:Alejandro Speck-Planche, Kleandrova V.V., Scotti M.T.Fuentes:scopus