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Development of Simplified Heterocyclic Acetogenin Analogues as Potent and Selective Trypanosoma brucei Inhibitors
ArticleAbstract: Neglected tropical diseases caused by parasitic infections are an ongoing and increasing concern. ThPalabras claves:Drug Discovery, natural product analogues, trypanosomatids, [3+2] cycloadditionAutores:Florence G.J., Fraser A.L., Gould E.R., King E.F.B., Morris J.C., Smith T.K., Stefanie K. Menzies, Thomson M.I., Tulloch L.B., Zacharova M.K.Fuentes:scopusNon-natural Acetogenin Analogues as Potent Trypanosoma brucei Inhibitors
ArticleAbstract: Neglected tropical diseases remain a serious global health concern. Here, a series of novel bis-tetrPalabras claves:acetogenin, Human African Trypanosomiasis (HAT), natural product analogues, Neglected diseases, stereochemistry, Trypanosoma bruceiAutores:Florence G.J., Fraser A.L., Gould E.R., King E.F.B., Morris J.C., Smith T.K., Stefanie K. Menzies, Tulloch L.B.Fuentes:scopus