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A putative antimicrobial peptide from Hymenoptera in the megaplasmid pSCL4 of Streptomyces clavuligerus ATCC 27064 reveals a singular case of horizontal gene transfer with potential applications
ArticleAbstract: Streptomyces clavuligerus is a Gram-positive bacterium that is a high producer of secondary metaboliPalabras claves:Antimicrobial peptide, horizontal gene transfer, Hymenoptera, pSCL4, Streptomyces clavuligerus ATCC 27064Autores:Daniela Santander-Gordón, Eduardo Tejera, Sebastián Ayala-Ruano, Vinicio Danilo Armijos-Jaramillo, Yunierkis Perez-CastilloFuentes:googlescopusTrypanocidal mechanism of action and in silico studies of p-coumaric acid derivatives
ArticleAbstract: Trypanosoma species are responsible for chronic and systemic infections in millions of people aroundPalabras claves:antiparasitic activity, cinnamic acid, esters, Natural products, Neglected diseases, Phenylpropanoid, TrypanosomaAutores:De Almeida R.N., de Menezes R.R.P.P.B., Lopes S.P., Martins A.M.C., Monteiro M.L., Sousa D.P.D., Yunierkis Perez-CastilloFuentes:googlescopusSynthetic Cinnamides and Cinnamates: Antimicrobial Activity, Mechanism of Action, and In Silico Study
ArticleAbstract: The severity of infectious diseases associated with the resistance of microorganisms to drugs highliPalabras claves:amides, Antimicrobial, Candida, cinnamic acid, esters, mechanism of action, Medicinal Plant, molecular docking, Natural product, S. AureusAutores:de Morais M.C., de Oliveira Lima E., Edeltrudes de Oliveira Lima, Sousa D.P.D., Yunierkis Perez-CastilloFuentes:googlescopusTI2BioP: Topological Indices to BioPolymers. Its practical use to unravel cryptic bacteriocin-like domains
ArticleAbstract: Bacteriocins are proteinaceous toxins produced and exported by both gram-negative and gram-positivePalabras claves:Alignment methods, Artificial secondary structure, Bacteriocin, Spectral moments, topological indicesAutores:Agüero-Chapin G., Antunes A., Molina-Ruiz R., Morales-Helguera A., Pérez-Machado G., Vasconcelos V., Yunierkis Perez-CastilloFuentes:googlescopusElucidating the Racemization Mechanism of Aliphatic and Aromatic Amino Acids by In Silico Tools
ArticleAbstract: The racemization of biomolecules in the active site can reduce the biological activity of drugs, andPalabras claves:amino acids, density functional theory, intrinsic reaction coordinates, Natural bond orbital, RacemizationAutores:Agüero-Chapin G., Andino M.S., José Luis Paz, Jose R. Mora, Marquez E.A., Yunierkis Perez-CastilloFuentes:scopusModeling defensive functions of alkaloids within diverse chemical portfolios
ReviewAbstract: Studies of the evolution of anti-predatory phenotypes such as aposematic signals have proven informaPalabras claves:alkaloids, Defenses, Defensive function, Modeling, Oophaga pumilio, Poison frogsAutores:Eduardo Tejera, Justin Yeager, Pablo Andres Viteri Chancusi, Vinicio Danilo Armijos-Jaramillo, Yunierkis Perez-CastilloFuentes:scopusCytotoxic and antifungal amides derived from ferulic acid: Molecular docking and mechanism of action
ArticleAbstract: Amides derived from ferulic acid have a wide spectrum of pharmacological activities, including antitPalabras claves:Autores:Bezerra D.P., De Castro R.D., de Morais M.C., de Souza Santos L., Silva V.R., Soares M.B.P., Sousa D.P.D., Yunierkis Perez-CastilloFuentes:googlescopusConsensus strategy in genes prioritization and combined bioinformatics analysis for preeclampsia pathogenesis
ArticleAbstract: Background: Preeclampsia is a multifactorial disease with unknown pathogenesis. Even when recent stuPalabras claves:Communality analysis, Consensus analysis, early recognition, Gene periodization, Microarray analysis, pathogenesis, PreeclampsiaAutores:Aminael Sánchez-Rodríguez, Borges F., Cesar Paz-y-Miño, Eduardo Tejera, Germán Burgos, Maykel Cruz-Monteagudo, Natalia Dias Soeiro Cordeiro M., Rebelo I., Sánchez M.E., Yunierkis Perez-CastilloFuentes:googlescopusArticle bioactive terpenes and their derivatives as potential SARS-CoV-2 proteases inhibitors from molecular modeling studies
ArticleAbstract: The coronavirus disease 2019 (COVID-19) pandemic is caused by a novel coronavirus; the Severe AcutePalabras claves:covid-19, MERS-CoV, Middle East Respiratory Syndrome Virus, Natural products, plants, saponins, SARS-CoV, SARS-CoV-2, Terpenoid, virusesAutores:Bezerra Filho C.d.S.M., Diniz L.R.L., Elshabrawy H.A., Sousa D.P.D., Yunierkis Perez-CastilloFuentes:googlescopusAntileishmanial Activity of Cinnamic Acid Derivatives against Leishmania infantum
ArticleAbstract: Leishmania infantum is the etiological agent of visceral leishmaniasis (VL) in South America, the MePalabras claves:antiparasitic activity, cinnamamide, cinnamate, Medicinal Plant, Natural productAutores:Almeida F.S., de Morais M.C., Gisele Alves Medeiros, Keesen T.d.S.L., Medeiros G.A., Rocha J.d.C., Sousa D.P.D., Yunierkis Perez-CastilloFuentes:googlescopus