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Comparative Study of Donepezil-Loaded Formulations for the Treatment of Alzheimer’s Disease by Nasal Administration
ArticleAbstract: Alzheimer’s disease is characterized by a progressive deterioration of neurons resulting in a steadyPalabras claves:Alzheimer’s disease, Donepezil, gel, intranasal administrationAutores:Brito-Llera A., Calpena A.C., Diana Guaya, Halbaut L., Lupe Carolina Espinoza, Mallandrich M., Perotti R.M., Sosa L.Fuentes:scopusComparative study of Ex Vivo transmucosal permeation of pioglitazone nanoparticles for the treatment of Alzheimer's disease
ArticleAbstract: Pioglitazone has been reported in the literature to have a substantial role in the improvement of ovPalabras claves:Alzheimer's disease, Nanoparticles, Pioglitazone, PLGA-PEG, Transmucosal permeationsAutores:Calpena A.C., Espina M., García M.L., Halbaut L., Lupe Carolina Espinoza, Silva-Abreu M.Fuentes:scopusApremilast microemulsion as topical therapy for local inflammation: Design, characterization and efficacy evaluation
ArticleAbstract: Apremilast (APR) is a selective phosphodiesterase 4 inhibitor administered orally in the treatment oPalabras claves:Apremilast, inflammation, Microemulsion, Phosphodiesterase 4, Skin DiseasesAutores:Badia J., Calpena A.C., Díaz-Garrido N., Fábrega M.J., Halbaut L., Lupe Carolina Espinoza, Paulo Sarango-Granda, Rodríguez-Lagunas M.J., Silva-Abreu M.Fuentes:scopusDevelopment of a nasal donepezil-loaded microemulsion for the treatment of Alzheimer’s disease: In vitro and Ex vivo characterization
ArticleAbstract: Background: Donepezil (DPZ) is widely prescribed as a specific and reversible acetylcholinesterase iPalabras claves:Alzheimer’s disease, Delivery systems, Donepezil, Intranasal route, Microemulsion, permeationAutores:Calpena A.C., Clares-Naveros B., Fábrega M.J., García M.L., Lupe Carolina Espinoza, Vacacela M.Fuentes:scopusFormulation strategies to improve nose-to-brain delivery of donepezil
ArticleAbstract: Donepezil (DPZ) is widely used in the treatment of Alzheimer’s disease in tablet form for oral adminPalabras claves:Alzheimer’s disease, Donepezil, Mucoadhesion, NANOEMULSIÓN, Nose-to-brain, Pluronic F-127Autores:Calpena A.C., Cañas M.A., Clares-Naveros B., Halbaut L., Lupe Carolina Espinoza, Rodríguez-Lagunas M.J., Silva-Abreu M.Fuentes:scopusQuality by Design of Pranoprofen Loaded Nanostructured Lipid Carriers and Their Ex Vivo Evaluation in Different Mucosae and Ocular Tissues
ArticleAbstract: Transmucosal delivery is commonly used to prevent or treat local diseases. Pranoprofen is an anti-inPalabras claves:design of experiment, nanostructured lipid carriers, ophthalmic tissues, permeation, porcine mucous membraneAutores:Abrego G., Calpena A.C., Lupe Carolina Espinoza, Mallandrich M., Pesantez-Narvaez J., Rincón M., Silva-Abreu M., Sosa L.Fuentes:scopusPolyene macrolide antibiotic nanoemulsion: a proposal for the treatment of cutaneous leishmaniasis
ArticleAbstract: Leishmaniasis is a neglected tropical disease that requires timely and inexpensive treatment. For thPalabras claves:Amphotericin B, Draize test, ex vivo permeation studies, histology, In vitro cytotoxicity, in vitro leishmanicidal activity, leishmaniasisAutores:Díaz M.R., Fuentes J.M., Lupe Carolina Espinoza, Rivas F.R., Siwady J.A., Sosa L.Fuentes:scopusNanoemulsion strategy of pioglitazone for the treatment of skin inflammatory diseases
ArticleAbstract: Pioglitazone (PGZ)is a peroxisome proliferator-activated receptor agonist. Its role in the inflammatPalabras claves:anti-inflammatory activity, cytokines, NANOEMULSIÓN, Pioglitazone, Skin disordersAutores:Calpena A.C., Clares-Naveros B., Fábrega M.J., Garduño-Ramírez M.L., Lupe Carolina Espinoza, Rodríguez-Lagunas M.J., Silva-Abreu M.Fuentes:scopusThiazolidinedione as an alternative to facilitate oral administration in geriatric patients with Alzheimer's disease
ArticleAbstract: Pioglitazone (PGZ) is a member of the thiazolidinedione (TZDs) family of drugs and it is primarily uPalabras claves:Alzheimer's disease, Geriatric patients, Mucosal permeation, Oral administration, Pioglitazone, ThiazolidinedionesAutores:Calpena A.C., Espina M., García M.L., Gonzalez-Pizarro R., Lupe Carolina Espinoza, Rodríguez-Lagunas M.J., Silva-Abreu M.Fuentes:scopusTopical pioglitazone nanoformulation for the treatment of atopic dermatitis: Design, characterization and efficacy in hairless mouse model
ArticleAbstract: Pioglitazone (PGZ) is a drug used to treat type 2 diabetes mellitus that has been reported to show aPalabras claves:Atopic dermatitis, NANOEMULSIÓN, Pioglitazone, Pluronic F127Autores:Badia J., Calpena A.C., Clares-Naveros B., Domènech Ò., Lupe Carolina Espinoza, Rodríguez-Lagunas M.J., Silva-Abreu M., Vera-García R.Fuentes:scopus