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scopus(16)
Synthesis of [60]Fullerene Hybrids Endowed with Steroids and Monosaccharides: Theoretical Underpinning as Promising anti-SARS-CoV-2 Agents
ArticleAbstract: Cyclopropanation reactions between C<inf>60</inf> and different malonates decorated with monosaccharPalabras claves:molecular docking, SARS-CoV-2, sugar steroid hybrids, Theoretical calculations, [60]FullereneAutores:Almagro L., Herranz M.Á., Hortensia Rodriguez Cabrera, Lemos R., Makowski K., Martín N., Molero D., Suárez Navarro M., Tolón B.Fuentes:scopusSynthesis of new carnitine palmitoyltransferase I inhibitors derivatives of C75
ArticleAbstract: Carnitine Palmitoyltransferase (CPT1) is an enzyme that catalyzes the transport of fatty acids fromPalabras claves:C75, Carnitine palmitoyltransferase 1 inhibitor, CPT1, α-Methylene-γ-butyrolactonesAutores:Alicia Venegas, Ariza J., Garcia J., Herrero L., Laura Herrero, Makowski K., Marta López, Mera P., Serra D.Fuentes:scopusTargeting energy expenditure—drugs for obesity treatment
ReviewAbstract: Obesity and overweight are associated with lethal diseases. In this context, obese and overweight inPalabras claves:clinical trials, energy expenditure, Energy metabolism, FDA-approved, obesity, Thermogenesis, Treatments under development, Withdrawn treatmentsAutores:Alberício F., Carlos M. Jimenez-Muñoz, Makowski K., Marta LópezFuentes:scopusSudemycin k: A synthetic antitumor splicing inhibitor variant with improved activity and versatile chemistry
ArticleAbstract: Important links exist between the process of pre-mRNA splicing and cancer, as illustrated by the frePalabras claves:Autores:Alberício F., Alvarez M., Juan Valcarcel, Luisa Vigevani, Makowski K.Fuentes:scopus[60]Fullerene Hybrids Bearing “Steroid Wings”: A Joined Experimental and Theoretical Investigation
ArticleAbstract: Novel [60]fullerene-steroid hybrids have been synthesized by Bingel–Hirsch cyclopropanation reactionPalabras claves:cyclopropanation, MORPHOLOGY, Steroid hybrids, Theoretical calculations, [60]FullereneAutores:Almagro L., Cáceres W., Herranz M.Á., Hortensia Rodriguez Cabrera, Lemos R., Makowski K., Martín N., Martínez-Álvarez R., Molero D., Ortiz O., Suárez Navarro M.Fuentes:scopusCrossed Aldol Reactions in Water Using Inexpensive and Easily Available Materials as a Tool for Reaction Optimization Teaching in an Undergraduate Organic Chemistry Laboratory
ArticleAbstract: We present an experiment designed to hone the decision-making skills of (undergraduate) chemistry stPalabras claves:Aqueous Solution Chemistry, Hands-On Learning/Manipulatives, organic chemistry, Problem Solving/Decision Making, Synthesis, Thin layer chromatographyAutores:Kevin A. Ruiz, Makowski K., Marta López, Suppan G.Fuentes:scopusAn Androsterone-H2@C60 hybrid: Synthesis, Properties and Molecular Docking Simulations with SARS-Cov-2
ArticleAbstract: We report the synthesis and characterization of a fullerene-steroid hybrid that contains H<inf>2</inPalabras claves:cyclopropanation, Fullerenes, molecular docking, SARS-CoV-2, Steroid hybridsAutores:Alberício F., Almagro L., Herranz M.Á., Hortensia Rodriguez Cabrera, Lemos R., Makowski K., Maroto E., Martín N., Molero D., Murata Y., Ortiz O., Suárez Navarro M.Fuentes:scopusInhibitors of lipogenic enzymes as a potential therapy against cancer
ReviewAbstract: Cancer cells rely on several metabolic pathways such as lipid metabolism to meet the increase in enePalabras claves:cancer drugs, lipid metabolism, lipogenic enzyme inhibitorsAutores:Ariza X., Herrero L., Laura Herrero, Makowski K., Marta López, Nicolás MontesdeocaFuentes:scopusNovel octapeptide containing the RGD sequence as a potential anti-SARS-CoV-2 agent: design, synthesis, and theoretical studies
ArticleAbstract: The design of peptide-based inhibitors targeting cell receptors represents a promising strategy in tPalabras claves:DFT calculations, Integrin α5β1, RGD motif, Solid-phase peptide synthesisAutores:Alberício F., Almagro L., Hortensia Rodriguez Cabrera, Makowski K., Ortiz O., Reiner Lemos, Suárez Navarro M.Fuentes:scopusDesign of new hybrids of fullerenes decorated with molecular fragments of chemical and biological relevance
ArticleAbstract: Introduction: In recent years, fullerenes have acquired great interest since their structure ena-blePalabras claves:Carbohydrates, cyclopropanation, Fullerenes, hybrid systems, steroidsAutores:Almagro L., Hortensia Rodriguez Cabrera, Lemos R., Makowski K., Martín N., Suárez Navarro M., Yoana Pérez-BadellFuentes:scopus