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Novel 7-Chloro-(4-thioalkylquinoline) Derivatives: Synthesis and Antiproliferative Activity through Inducing Apoptosis and DNA/RNA Damage
ArticleAbstract: A series of 78 synthetic 7-chloro-(4-thioalkylquinoline) derivatives were investigated for cytotoxicPalabras claves:antiproliferative activity, cell cycle, DNA/RNA damage, Sulfanyl-Sulfinyl-Sulfonyl groups, synthesis of 4-thioalkylquinolineAutores:Bruno-Colmenarez J., Charris J.E., de Sanctis J.B., Deffieux D., Džubák P., Esteban Fernández-Moreira, Gurská S., Gutiérrez J.E., Hajdůch M., Hegira Ramírez, Mijares M.R., Pouységu L., Quideau S., Rodríguez M.A., Rojas L.B.Fuentes:scopusOne-pot multicomponent synthesis of methoxybenzo[h]quinoline-3-carbonitrile derivatives; anti-chagas, X-ray, and in silico ADME/tox profiling studies
ArticleAbstract: Several methoxybenzo[h]quinoline-3-carbonitrile analogs were designed and synthesized in a repositioPalabras claves:Cáncer, chagas, Methoxybenzo[h]quinoline, One-pot synthesisAutores:Ángel J.E., Capparelli M.V., Charris J.E., Charris K.E., Esteban Fernández-Moreira, Hegira Ramírez, Nogueda-Torres B.Fuentes:scopusSYNTHESIS OF 4-BENZYLSULFANYL AND 4-BENZYLSULFONYL CHALCONES. BIOLOGICAL EVALUATION AS ANTIMALARIAL AGENTS
ArticleAbstract: Malaria management has been complicated in recent times, perhaps, by increasing the Plasmodium spp.Palabras claves:Antimalarial, Chalcones, Plasmodium berghei, β-haematinAutores:Charris J.E., Domínguez J.N., Esteban Fernández-Moreira, Hegira Ramírez, Rodrigues J.R., Rodríguez M.A.Fuentes:scopusSynthesis, Leishmanicidal, Trypanocidal, Antiproliferative Assay and Apoptotic Induction of (2-Phenoxypyridin-3-yl)naphthalene-1(2H)-one Derivatives
ArticleAbstract: The coexistence of leishmaniasis, Chagas disease, and neoplasia in endemic areas has been extensivelPalabras claves:apoptosis, Cáncer, chalcone, leishmaniasis, TRYPANOSOMA CRUZIAutores:Ángel J.E., Blanco Z., Celis C., Charris J.E., de Sanctis J.B., Džubák P., Esteban Fernández-Moreira, García Y., Gurská S., Hajdůch M., Hegira Ramírez, Jhonny Correa-Abril, Martinez G.P., Mijares M.R., Mijoba A., Nahum Herrera, Serrano X., Yonathan De J. ParraFuentes:scopusSynthesis, dopaminergic profile, and molecular dynamics calculations of N-aralkyl substituted 2-aminoindans
ArticleAbstract: Brain dopaminergic system has a crucial role in the etiology of several neuropsychiatric disorders,Palabras claves:Apomorphine-stereotypy, dopamine, molecular dynamics simulations, N-Aralkyl 2-aminoindan derivativesAutores:Andujar S.A., Angel-Guío J.E., Charris J.E., de Angel B.M., Elvia V. Cabrera-Maldonado, Enriz R.D., Garrido M.R., Israel A., López S.E., Rosales C., Suárez-Roca H., Suvire F.D., Visbal G.Fuentes:scopus