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Conformation-dependent QSAR approach for the pbkp_rediction of inhibitory activity of bromodomain modulators
ArticleAbstract: Epigenetic drug discovery is a promising research field with growing interest in the scientific commPalabras claves:3D molecular descriptors, Applicability domain, Bromodomains, epigenetic drug discovery, QSAR, QuBiLS-MIDAS, ToMoCoMD-CARDDAutores:César R. García-Jacas, Martinez-Mayorga K., Medina-Franco J.L., Yovani Marrero-PonceFuentes:scopusSynthesis, anti-inflammatory activity and modeling studies of cycloartane-type terpenes derivatives isolated from Parthenium argentatum
ArticleAbstract: The 12-O-tetradecanoylphorbol-13-acetate (TPA)-induced edema model in mice determined the anti-inflaPalabras claves:anti-inflammatory activity, Argentatins, Cycloartanes, docking, TPA-induced mice model, TriterpenesAutores:Herrera M.P., Juan Carlos Romero-Benavides, Martinez-Mayorga K., Martínez-Vázquez A., Martínez-Vázquez M., Parra-Delgado H., Pérez-Flores F.J.Fuentes:googlescopus