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Effect of α-Methoxy Substitution on the Anti-HIV Activity of Dihydropyrimidin-4(3 H)-ones
ArticleAbstract: Conformational restriction applied to dihydrobenzylpyrimidin-4-(3H)-ones (DABOs) by the intoductionPalabras claves:Autores:Badia R., Cirilli R., Crespan E., Esté J.A., Forgione M., Hailu G., Jorge I. Armijos-Rivera, Kirillov I., Lucidi A., Maga G., Mai A., Nawrozkij M., Panella C., Patsilinakos A., Ragno R., Riveira-Munoz E., Rotili D., Tomaselli D., Yablokov A.Fuentes:googlescopusNew indolylarylsulfone non-nucleoside reverse transcriptase inhibitors show low nanomolar inhibition of single and double HIV-1 mutant strains
ArticleAbstract: We designed and synthesized 21 new indolylarylsulfones (IASs) as new HIV-1 NNRTIs. Among these, IASPalabras claves:AIDs, HIV-1, Indolylarylsulfone, Non-nucleoside reverse transcriptase inhibitor, Reverse transcriptaseAutores:Badia R., Brambilla A., Catalano M., Cinquina E., Coluccia A., Crespan E., Esté J.A., Falasca F., Jorge I. Armijos-Rivera, La Regina G., Limatola C., Maga G., Masci D., Nalli M., Riveira-Munoz E., Silvestri R., Turriziani O.Fuentes:scopus