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SYNTHESIS OF 4-BENZYLSULFANYL AND 4-BENZYLSULFONYL CHALCONES. BIOLOGICAL EVALUATION AS ANTIMALARIAL AGENTS
ArticleAbstract: Malaria management has been complicated in recent times, perhaps, by increasing the Plasmodium spp.Palabras claves:Antimalarial, Chalcones, Plasmodium berghei, β-haematinAutores:Charris J.E., Domínguez J.N., Esteban Fernández-Moreira, Hegira Ramírez, Rodrigues J.R., Rodríguez M.A.Fuentes:scopusSynthesis and antimalarial and anticancer evaluation of 7-chlorquinoline-4-thiazoleacetic derivatives containing aryl hydrazide moieties
ArticleAbstract: Twelve 7-chloroquinoline derivatives were designed and synthesized using the principle of molecularPalabras claves:Antimalarial, Antiproliferative, apoptosis, hydrazides, quinoline, thiazolAutores:Celis C., Charris J.E., de Sanctis J.B., Esteban Fernandez, Hegira Ramírez, Martinez G.P., Mayora S., Mijares M.R., Rodrigues J.R.Fuentes:scopusSynthesis and biological activity of 2-[2-(7-chloroquinolin-4-ylthio)-4-methylthiazol-5-yl]-N-phenylacetamide derivatives as antimalarial and cytotoxic agents
ArticleAbstract: A novel series of 2-[2-(7-chloroquinolin-4-ylthio)-4-methylthiazol-5-yl]-N-phenylacetamide derivativPalabras claves:ANTICANCER, Antimalarial, plasmodium, quinoline, thiazoleacetic acidAutores:Charris J.E., de Sanctis J.B., Hegira Ramírez, Mijares M.R., Rodrigues J.R.Fuentes:scopus