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A2AR transmembrane 2 peptide administration disrupts the A2AR-A2AR homoreceptor but not the A2AR-D2R heteroreceptor complex: Lack of actions on rodent cocaine self-administration
ArticleAbstract: It was previously demonstrated that rat adenosine A2AR transmembrane V peptide administration into tPalabras claves:Adenosine A2A receptor, Allosteric receptor–receptor interactions, cocaine use disorder, dopamine D2 receptor, Heteroreceptor complexes, Homoreceptor complexes, Small interfering peptides: G protein-coupled receptorsAutores:Borroto-Escuela D.O., Filip M., Frankowska M., Fuxe K., W. Romero-Fernandez, Wydra K., Zhou Z.Fuentes:scopusOSU-6162, a Sigma1R Ligand in Low Doses, Can Further Increase the Effects of Cocaine Self-Administration on Accumbal D2R Heteroreceptor Complexes
ArticleAbstract: Cocaine was previously shown to act at the Sigma1R which is a target for counteracting cocaine actioPalabras claves:A2AR-D2R heteroreceptor complexes, allosteric receptor-receptor interactions, cocaine use disorder, monoamine stabilizerAutores:Borroto-Escuela D.O., Filip M., Fuxe K., Suder A., W. Romero-Fernandez, Wydra K., Zhou Z.Fuentes:scopus