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A2AR transmembrane 2 peptide administration disrupts the A2AR-A2AR homoreceptor but not the A2AR-D2R heteroreceptor complex: Lack of actions on rodent cocaine self-administration
ArticleAbstract: It was previously demonstrated that rat adenosine A2AR transmembrane V peptide administration into tPalabras claves:Adenosine A2A receptor, Allosteric receptor–receptor interactions, cocaine use disorder, dopamine D2 receptor, Heteroreceptor complexes, Homoreceptor complexes, Small interfering peptides: G protein-coupled receptorsAutores:Borroto-Escuela D.O., Filip M., Frankowska M., Fuxe K., W. Romero-Fernandez, Wydra K., Zhou Z.Fuentes:scopusAcute cocaine treatment enhances the antagonistic allosteric adenosine A2A-dopamine D2 receptor–receptor interactions in rat dorsal striatum without increasing significantly extracellular dopamine levels
ArticleAbstract: Background: Antagonistic adenosine A2A receptor (A2AR)-dopamine D2 receptor (D2R) receptor–receptorPalabras claves:Adenosine A2A receptor, Cocaine, dopamine D2 receptor, Heteroreceptor complexes, Sigma1 receptorAutores:Beggiato S., Borroto-Escuela D.O., Ferraro L., Filip M., Fuxe K., Tanganelli S., W. Romero-Fernandez, Wydra K., Zhou Z.Fuentes:scopusOSU-6162, a Sigma1R Ligand in Low Doses, Can Further Increase the Effects of Cocaine Self-Administration on Accumbal D2R Heteroreceptor Complexes
ArticleAbstract: Cocaine was previously shown to act at the Sigma1R which is a target for counteracting cocaine actioPalabras claves:A2AR-D2R heteroreceptor complexes, allosteric receptor-receptor interactions, cocaine use disorder, monoamine stabilizerAutores:Borroto-Escuela D.O., Filip M., Fuxe K., Suder A., W. Romero-Fernandez, Wydra K., Zhou Z.Fuentes:scopusIncreased density and antagonistic allosteric interactions in A2AR-D2R heterocomplexes in extinction from cocaine use, lost in cue induced reinstatement of cocaine seeking
ArticleAbstract: Neurochemical studies were previously performed on the effects of a 10 day extinction learning fromPalabras claves:Adenosine A2A receptor, Cocaine extinction, Cocaine self-administration, dopamine D2 receptor, G protein-coupled receptors, Heteroreceptor complexes, Substance use disorderAutores:Borroto-Escuela D.O., Filip M., Frankowska M., Fuxe K., Jastrzębska J., W. Romero-Fernandez, Wydra K., Zhou Z.Fuentes:scopus