Siverio-Mota D.
53
Coauthors
5
Documentos
Volumen de publicaciones por año
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Año de publicación | Num. Publicaciones |
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2011 | 1 |
2013 | 2 |
2017 | 2 |
Publicaciones por áreas de conocimiento
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Área de conocimiento | Num. Publicaciones |
---|---|
Farmacología | 7 |
Descubrimiento de fármacos | 3 |
Bioquímica | 1 |
Biotecnología | 1 |
Publicaciones por áreas temáticas
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Área temática | Num. Publicaciones |
---|---|
Farmacología y terapéutica | 4 |
Química y ciencias afines | 2 |
Medicina y salud | 1 |
Bioquímica | 1 |
Microorganismos, hongos y algas | 1 |
Principales fuentes de datos
Origen | Num. Publicaciones |
---|---|
Scopus | 5 |
RRAAE | 2 |
Google Scholar | 1 |
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Coautores destacados por número de publicaciones
Coautor | Num. Publicaciones |
---|---|
Crawford A.D. | 5 |
De Witte P.A.M. | 5 |
María Lorena Cordero-Maldonado | 4 |
Vicet-Muro L. | 3 |
Yovani Marrero-Ponce | 3 |
Arán V.J. | 3 |
Giner R.M. | 3 |
Esguerra C.V. | 3 |
Veítia M.S.I. | 2 |
Pérez-Jiménez F. | 1 |
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Publicaciones del autor
Optimization and Pharmacological Validation of a Leukocyte Migration Assay in Zebrafish Larvae for the Rapid In Vivo Bioactivity Analysis of Anti-Inflammatory Secondary Metabolites
ArticleAbstract: Over the past decade, zebrafish (Danio rerio) have emerged as an attractive model for in vivo drug dPalabras claves:Autores:Crawford A.D., De Witte P.A.M., Esguerra C.V., Isabel María Wilches Arizabala, María Lorena Cordero-Maldonado, Siverio-Mota D., Vicet-Muro L., Wilches IsabelFuentes:rraaescopusDiscovery of novel anti-inflammatory drug-like compounds by aligning in silico and in vivo screening: The nitroindazolinone chemotype
ArticleAbstract: In this report, we propose the combination of computational methods and in vivo primary screening inPalabras claves:Anti-inflammatory compound, Anti-inflammatory database, Atom-based quadratic indices, Computational Screening, Cytotoxicity, In vivo anti-inflammatory assay, lead generation, Learning machine-based QSAR, ToMoCoMD-CARDD software, zebrafishAutores:Arán V.J., Crawford A.D., De Witte P.A.M., Esguerra C.V., Gálvez-Llompart M., García-Domnech R., Giner R.M., María Lorena Cordero-Maldonado, Recio M.C., Siverio-Mota D., Torrens F., Yovani Marrero-PonceFuentes:scopusIntegration of Microfractionation, qNMR and Zebrafish Screening for the In Vivo Bioassay-Guided Isolation and Quantitative Bioactivity Analysis of Natural Products
ArticleAbstract: Natural products (NPs) are an attractive source of chemical diversity for small-molecule drug discovPalabras claves:Autores:Bohni N., Crawford A.D., De Witte P.A.M., Esguerra C.V., Kamuhabwa A.R., Maes J., Marcourt L., María Lorena Cordero-Maldonado, Moshi M.J., Munck S., Siverio-Mota D., Wolfender J.L.Fuentes:rraaescopusAnti-inflammatory activity and cheminformatics analysis of new potent 2-substituted 1-methyl-5-nitroindazolinones
ArticleAbstract: After the identification of the anti-inflammatory properties of VA5-13l (2-benzyl-1- methyl-5-nitroiPalabras claves:Anti-inflammatory compound, Nitroindazolinones, SARANEA software, Structure-activity relationship, TPA-induced mouse ear edema, zebrafishAutores:Andújar I., Arán V.J., Crawford A.D., De Witte P.A.M., Díaz-Mendoza C., Giner R.M., Manjarrez G., María Lorena Cordero-Maldonado, Pérez-Jiménez F., Siverio-Mota D., Veítia M.S.I., Vicet-Muro L., Yovani Marrero-PonceFuentes:scopusFishing anti-inflammatories from known drugs: In silico repurposing, design, synthesis and biological evaluation of bisacodyl analogues
ArticleAbstract: Herein is described in silico repositioning, design, synthesis, biological evaluation and structure-Palabras claves:Anti-inflammatory assay, Anti-inflammatory database, Atom-based bilinear indices, Bisacodyl, Diarylmethylpyridines, Repurposing, ToMoCoMD-CARDD softwareAutores:Arán V.J., Crawford A.D., De Witte P.A.M., Dumas F., Ferroud C., Giner R.M., Guerra Y.R., Lerari V., Marín M., Siverio-Mota D., Veítia M.S.I., Vicet-Muro L., Yovani Marrero-PonceFuentes:googlescopus