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4-Aryl(benzyl)amino-4-heteroarylbut-1-enes as building blocks in heterocyclic synthesis. 4.<sup>1</sup> synthesis of 4,6-dimethyl-5-nitro(amino)- 2-pyridylquinolines and their antiparasitic activities
ArticleAbstract: New nitro- and aminoquinoline derivatives containing a pyridyl nucleus were synthesized from 6,8-disPalabras claves:Aminoquinolines, Antichagasic, Cytotoxic properties, Nitroquinolines, TrichomonacidalAutores:Bahsas A., Fernández Portillo C., Gómez-Barrio A., Juan Manuel Amaro-Luis, Kouznetsov V.V., Montero Pereira D., Muelas Serrano S., Nogal-Ruiz J.J., Ochoa C., Tibaduiza B., Vargas Méndeź L.Y.Fuentes:scopusA linear discrimination analysis based virtual screening of trichomonacidal lead-like compounds: Outcomes of in silico studies supported by experimental results
ArticleAbstract: A computational (virtual) screening test to identify potential trichomonacidals has been developed.Palabras claves:Atom-based quadratic indices, Cytotoxic properties, LDA-based model, ToMoCoMD-CARDD software, TrichomonacidalAutores:Arán V.J., García-Sánchez R.N., García-Trevijano J.A.E., Machado-Tugores Y., Martínez-Fernández A.R., Meneses-Marcel A., Montero-Torres A., Nogal-Ruiz J.J., Ochoa C., Pereira D.M., Yovani Marrero-PonceFuentes:googlescopus