Documentos de Monaim S.A.H.A. | REDI

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Mostrando 10 resultados de: 10

Subtipo de publicación

Publisher

Bioorganic and Medicinal Chemistry(1)

Frontiers in Microbiology(1)

Área temáticas

Farmacología y terapéutica(8)

Microorganismos, hongos y algas(4)

Química orgánica(4)

Área de conocimiento

Microbiología(2)

Resistencia antimicrobiana(2)

Antibiótico(1)

Año de Publicación

Origen

Palabras Claves

Solid-phase peptide synthesis(4)

Antimicrobial peptides(2)

biological activity(2)

cyclic peptides(2)

Bacteria Hunt Bacteria through an Intriguing Cyclic Peptide

Abstract: In the last few decades, peptides have been victorious over small molecules as therapeutics due to t

Palabras claves:

Antibiotics, biological activity, cyclic antimicrobial peptides, Drug Discovery, Peptides

Alberício F., B. G. De la Torre, El-Faham A., Monaim S.A.H.A., Somboro A.M.

Converting Teixobactin into a Cationic Antimicrobial Peptide (AMP)

Abstract: Teixobactin is a head to side chain cyclodepsipeptide that contains two positive charges. One is fou

Palabras claves:

Alberício F., B. G. De la Torre, El-Faham A., Monaim S.A.H.A., Ramchuran E.J.

Formation of N <sup>α</sup>-terminal 2-dialkyl amino oxazoles from guanidinated derivatives under mild conditions

Abstract: Oxazole-containing peptides are an important class of molecules in medicinal chemistry programs. Her

Palabras claves:

Alberício F., B. G. De la Torre, El-Faham A., Kumar A., Mhlongo J.T., Monaim S.A.H.A.

N-methylation in amino acids and peptides: Scope and limitations

Abstract: Active pharmaceutical ingbkp_redients (APIs) can be divided into two types, namely chemical and biol

Palabras claves:

cyclic peptides, NMAA, side-reactions, Solid-phase peptide synthesis

Alberício F., B. G. De la Torre, El-Faham A., Jad Y.E., Kumar A., Monaim S.A.H.A., Sharma A.

In vitro antibacterial activity of Teixobactin derivatives on clinically relevant bacterial isolates

Abstract: Methicillin-resistant Staphylococcus aureus (MRSA) and vancomycin-resistant enterococcus (VRE) are i

Palabras claves:

Antimicrobial agents, Antimicrobial peptides, biological activity, in silico analysis, resistant bacteria, Teixobactin derivatives

Agrawal N., Alberício F., Amoako D.G., B. G. De la Torre, Bester L.A., Kumalo H.M., Monaim S.A.H.A., Parboosing R., Ramchuran E.J., Somboro A.M.

Lysine scanning of Arg<inf>10</inf>−teixobactin: Deciphering the role of hydrophobic and hydrophilic residues

Abstract: Teixobactin is a recently discovered antimicrobial cyclodepsipeptide with good activity against Gram

Palabras claves:

Alberício F., B. G. De la Torre, El-Faham A., Govender T., Jad Y.E., Kruger H.G., Monaim S.A.H.A., Ramchuran E.J.

Investigation of the N-terminus amino function of Arg<inf>10</inf>-Teixobactin

Abstract: Teixobactin is a recently described antimicrobial peptide that shows high activity against gram-posi

Palabras claves:

Antimicrobial peptides, Cyclic depsipeptides, Lipophilicity, Solid-phase peptide synthesis, Teixobactin

Alberício F., B. G. De la Torre, El-Faham A., Monaim S.A.H.A., Noki S., Ramchuran E.J.

Re-evaluation of the N-terminal substitution and the D-residues of teixobactin

Abstract: Teixobactin is a head to side-chain cyclic depsipeptide with a guanidino based residue within the cy

Palabras claves:

Acosta G.A., Alberício F., B. G. De la Torre, El-Faham A., Govender T., Jad Y.E., Kruger H.G., Monaim S.A.H.A., Naicker T., Ramchuran E.J.

Solid-phase synthesis of homodetic cyclic peptides from Fmoc-MeDbz-resin

Abstract: Cyclic homodetic peptides are very appealing for medicinal chemistry programs. In addition to the hi

Palabras claves:

Cyclactive cleavage, cyclic peptides, MeDbz linker, Solid-phase peptide synthesis

Acosta G.A., Alberício F., B. G. De la Torre, El-Faham A., Monaim S.A.H.A., Royo M.

Teixobactin as a scaffold for unlimited new antimicrobial peptides: SAR study

Abstract: It looks that a new era of antimicrobial peptides (AMPs) started with the discovery of teixobactin,

Palabras claves:

Antimicrobial Resistance, cyclic peptide, Depsipeptide, Gram-positive bacteria, Solid-phase peptide synthesis

Alberício F., B. G. De la Torre, El-Faham A., Jad Y.E., Monaim S.A.H.A.