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Article(2)
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Abiraterone inhibits 3β-hydroxysteroid dehydrogenase: A rationale for increasing drug exposure in castration-resistant prostate cancer
ArticleAbstract: Purpose: Treatment with abiraterone (abi) acetate prolongs survival in castration-resistant prostatePalabras claves:Autores:Chang K.H., Evaul K., Li R., Liu J., Richard J. Auchus, Sharifi N., Sharma K.K., Yoshimoto J.A.Fuentes:scopusSelectivity of osilodrostat as an inhibitor of human steroidogenic cytochromes P450
ArticleAbstract: Osilodrostat (LCI699) is a potent inhibitor of the human steroidogenic cytochromes P450 11β-hydroxylPalabras claves:Cushing syndrome, Cytochrome p450, LCI699, Osilodrostat, steroidogenesisAutores:Liu J., Oommen J., Peng H.M., Richard J. Auchus, Valentín-Goyco J.Fuentes:scopus