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Article(5)
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Journal of Steroid Biochemistry and Molecular Biology(2)
Endocrinology (United States)(1)
Nature(1)
Nature Communications(1)
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Bioquímica(2)
Farmacología y terapéutica(2)
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Microorganismos, hongos y algas(1)
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Bioquímica(3)
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Cáncer(1)
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ODS 3: Salud y bienestar(5)
ODS 10: Reducción de las desigualdades(4)
ODS 6: Agua limpia y saneamiento(1)
Origen
scopus(5)
Conversion of abiraterone to D4A drives anti-tumour activity in prostate cancer
ArticleAbstract: Prostate cancer resistance to castration occurs because tumours acquire the metabolic capability ofPalabras claves:Autores:Alyamani M., Bishop A., Bunch D., Dreicer R., Garcia J., Li Z., Liu J., Richard J. Auchus, Sharifi N., Upadhyay S.K.Fuentes:scopusFunctional characterization of the G162R and D216H genetic variants of human CYP17A1
ArticleAbstract: Cytochrome P450 17A1 (CYP17A1) is a dual-function enzyme catalyzing reactions necessary for cortisolPalabras claves:CYP17A1, Cytochrome p450, Proteasome, steroidogenesis, UbiquitinationAutores:Capper C.P., Hollenberg P.F., Johnson M.D., Larios J.M., Liu J., McIntosh L.R., Osawa Y., Rae J.M., Richard J. AuchusFuentes:scopusExpression in escherichia coli, purification, and functional reconstitution of human steroid 5α-reductases
ArticleAbstract: The potent androgen 5α-dihydrotestosterone irreversibly derives from testosterone via the activity oPalabras claves:5α-reductase, androgen, Dihydrotestosterone, prostate, steroidogenesisAutores:Han B., Im S.C., Liu J., Peng H.M., Qiao J., Richard J. Auchus, Valentín-Goyco J.Fuentes:scopusSelectivity of osilodrostat as an inhibitor of human steroidogenic cytochromes P450
ArticleAbstract: Osilodrostat (LCI699) is a potent inhibitor of the human steroidogenic cytochromes P450 11β-hydroxylPalabras claves:Cushing syndrome, Cytochrome p450, LCI699, Osilodrostat, steroidogenesisAutores:Liu J., Oommen J., Peng H.M., Richard J. Auchus, Valentín-Goyco J.Fuentes:scopusMaking water-soluble integral membrane proteins in vivo using an amphipathic protein fusion strategy
ArticleAbstract: Integral membrane proteins (IMPs) play crucial roles in all cells and represent attractive pharmacolPalabras claves:Autores:Chen Y., Delisa M.P., Ke A., Liu J., Mizrachi D., Peng H.M., Pollack L., Richard J. Auchus, Turner R.J.Fuentes:scopus