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Anti-Cancer Agents in Medicinal Chemistry(1)
Bioorganic and Medicinal Chemistry(1)
Current Alzheimer Research(1)
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scopus(5)
Chemoinformatics for rational discovery of safe antibacterial drugs: Simultaneous pbkp_redictions of biological activity against streptococci and toxicological profiles in laboratory animals
ArticleAbstract: Streptococci are a group of Gram-positive bacteria which are responsible for causing many diverse diPalabras claves:antibacterial, Artificial neural network mtk-QSAR, Streptococci, topological indicesAutores:Alejandro Speck-Planche, Kleandrova V.V., Natalia Dias Soeiro Cordeiro M.Fuentes:scopusMulti-target inhibitors for proteins associated with Alzheimer: In silico discovery using fragment-based descriptors
ArticleAbstract: Alzheimer disease (AD) is one of the most common and serious neurodegenerative disorders in humans.Palabras claves:Anti-AD agents, Fragment, linear discriminant analysis, Mt-inhibitors, QSAR, quantitative contributionsAutores:Alejandro Speck-Planche, Kleandrova V.V., Luan F., Natalia Dias Soeiro Cordeiro M.Fuentes:scopusUnified multi-target approach for the rational in silico design of anti-bladder cancer agents
ArticleAbstract: Bladder cancer (BLC) is a very dangerous and common disease which is characterized by an uncontrollePalabras claves:artificial neural networks, bladder cancer, Fragments, In silico design, linear discriminant analysis, Molecular descriptors, Mt- QSAR, quantitative contributionsAutores:Alejandro Speck-Planche, Kleandrova V.V., Luan F., Natalia Dias Soeiro Cordeiro M.Fuentes:scopusThe latest guidance on the simultaneous design of virtually active and non-hemolytic peptides
OtherAbstract:Palabras claves:activity, design, hemotoxicity, peptide, PTML, topological indicesAutores:Alejandro Speck-Planche, Kleandrova V.V.Fuentes:scopusThe urgent need for pan-antiviral agents: From multitarget discovery to multiscale design
ReviewAbstract:Palabras claves:COVID-19 •drug repurposing, multiscale de novo drug design, multitarget inhibitor, new molecular entity, pan-antiviral, PTML, SARS-COV-2Autores:Alejandro Speck-Planche, Kleandrova V.V.Fuentes:scopus