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scopus(8)
Di- and tri-substituted s-triazine derivatives: Synthesis, characterization, anticancer activity in human breast-cancer cell lines, and developmental toxicity in zebrafish embryos
ArticleAbstract: Here we report on a small library based on a 4-aminobenzonitile-s-triazine moiety. We used a straighPalabras claves:4-aminobenzonitile-s-triazine, anticancer activity, Di- trisubstituted s-triazine, Zebrafish embryosAutores:Alberício F., Alhameed R.A., Almarhoon Z.M., B. G. De la Torre, El-Faham A., Farooq M., Wadaan M.A.M.Fuentes:scopusDesign and synthesis of mono-and di-pyrazolyl-s-triazine derivatives, their anticancer profile in human cancer cell lines, and in vivo toxicity in zebrafish embryos
ArticleAbstract: s-Triazine is considered a privileged structure, as it is found in several FDA-approved drugs. In thPalabras claves:anticancer activity, Pyrazole, S-triazine, Zebrafish embryosAutores:Al-Dhfyan A., Alberício F., Almarhoon Z.M., B. G. De la Torre, El-Faham A., Farooq M., Sharma A., Taha N.A., Wadaan M.A.M.Fuentes:scopusExploiting the Thiobarbituric Acid Scaffold for Antibacterial Activity
ArticleAbstract: Thiobarbituric acid (TBA) has been considered a privileged structure for developing antimicrobial agPalabras claves:Antibiotics, barbituric acid, nanoformulations, Thiobarbituric acidAutores:Alberício F., Almarhoon Z.M., B. G. De la Torre, El-Faham A., Hazzah H.A., Noki S., Sharma A., Zamisa S.J.Fuentes:scopusNovel 4,6-disubstituted s-triazin-2-yl amino acid derivatives as promising antifungal agents
ArticleAbstract: A novel series of 4,6-disubstituted s-triazin-2-yl amino acid derivatives was prepared and characterPalabras claves:2,4,6-trichlorotriazine, Antifungal, Candida Albicans, N-myristoltransferase, TCT, Triazine amino acidAutores:Alberício F., Alhameed R.A., Almarhoon Z.M., B. G. De la Torre, El-Faham A., Khan S.A., Sharma A., Sholkamy E.N., Ul-Haq Z.Fuentes:scopusNutraceutical Profiling, Bioactive Composition, and Biological Applications of Lepidium sativum L.
ReviewAbstract: The roots, leaves, and seeds of Lepidium sativum L., popularly known as Garden cress in different rePalabras claves:Autores:Almarhoon Z.M., Alshehri M.M., Calina D., Cho W.C., Daştan S.D., Herrera-Bravo J., Javad Sharifi Rad, Martorell M., Painuli S., Quispe C., Seilkhan A., Semwal P., Taheri Y., Ydyrys A.Fuentes:scopusProtocol for synthesis of di- and tri-substituted s-triazine derivatives
ArticleAbstract: The present protocol describes the synthesis of di and tri-substituted s-triazine derivatives • s-TrPalabras claves:ALCOHOL, amines, Cyanuric chloride, Nucleophilic substitution, Orthogonal chemoselectivity, Sequential nucleophilic substitutionAutores:Alberício F., Alhameed R.A., Almarhoon Z.M., B. G. De la Torre, El-Faham A., Farooq M., Sharma A., Wadaan M.A.M.Fuentes:scopusSynthesis and antimicrobial activity of a new series of thiazolidine-2,4-diones carboxamide and amino acid derivatives
ArticleAbstract: Novel thiazolidine-2,4-dione carboxamide and amino acid derivatives were synthesized in excellent yiPalabras claves:Antibacterial activity, OxymaPure, Thiazolidine-2,4-dione amino acid ester, Thiazolidine-2,4-dione carboxamideAutores:Alberício F., Alhameed R.A., Almarhoon Z.M., B. G. De la Torre, Bukhari S.I., El-Faham A.Fuentes:scopusThe antiproliferative and apoptotic effect of a novel synthesized s-triazine dipeptide series, and toxicity screening in zebrafish embryos
ArticleAbstract: Several derivatives containing morpholine/piperidine, anilines, and dipeptides as pending moieties wPalabras claves:Anti-proliferative activity, apoptosis, Dipeptides, S-triazine, zebrafishAutores:Alberício F., Alhameed R.A., Almarhoon Z.M., B. G. De la Torre, El-Faham A., Farooq M., Malebari A.M., Sharma A., Wadaan M.A.M.Fuentes:scopus