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scopus(34)
Barbiturate- And Thiobarbituarte-Based s-Triazine Hydrazone Derivatives with Promising Antiproliferative Activities
ArticleAbstract: A new class of compounds, which include s-triazine with pyrimidinetrione or thiopyrimidinedione moiePalabras claves:Autores:Al-Rasheed H.H., Alberício F., B. G. De la Torre, Dahlous K.A., El-Faham A., Sharma A., Sholkamy E.N.Fuentes:scopus1,3,5-Triazino Peptide Derivatives: Synthesis, Characterization, and Preliminary Antileishmanial Activity
ArticleAbstract: A library of short di-, tri-, and tetra-peptides with an s-triazine moiety at the N terminus and eitPalabras claves:1,3,5-triazine derivatives, antileishmanial compounds, morpholines, Peptides, piperidinesAutores:Abd El-Rahman M.M., Alberício F., B. G. De la Torre, Bekhit A.A., El-Faham A., Khalil H.H., Khattab S.N.Fuentes:scopusDi- and tri-substituted s-triazine derivatives: Synthesis, characterization, anticancer activity in human breast-cancer cell lines, and developmental toxicity in zebrafish embryos
ArticleAbstract: Here we report on a small library based on a 4-aminobenzonitile-s-triazine moiety. We used a straighPalabras claves:4-aminobenzonitile-s-triazine, anticancer activity, Di- trisubstituted s-triazine, Zebrafish embryosAutores:Alberício F., Alhameed R.A., Almarhoon Z.M., B. G. De la Torre, El-Faham A., Farooq M., Wadaan M.A.M.Fuentes:scopusConverting Teixobactin into a Cationic Antimicrobial Peptide (AMP)
ArticleAbstract: Teixobactin is a head to side chain cyclodepsipeptide that contains two positive charges. One is fouPalabras claves:Autores:Alberício F., B. G. De la Torre, El-Faham A., Monaim S.A.H.A., Ramchuran E.J.Fuentes:scopusCorrigendum: Pyrazolyl-s-triazine with indole motif as a novel of epidermal growth factor receptor/cyclin-dependent kinase 2 dual inhibitors(Front. Chem., (2022), 10, (1078163), 10.3389/fchem.2022.1078163)
OtherAbstract: In the original article, there was an error in the Affiliation for Samha Al Ayoubi2. Instead of “SamPalabras claves:anticancer profile, apoptosis, EGFR/CDK-2, ÍNDOLE, pyrazolyl-s-triazineAutores:Al Ayoubi S., Al Zoubi M., Al-Rasheed H.H., Alberício F., Aldalbahi A., Ali M., Alshaer W., B. G. De la Torre, Barakat A., El-Faham A., Nafie M.S., Shawish I.Fuentes:scopusAcetic Acid Mediated for One-Pot Synthesis of Novel Pyrazolyl s-Triazine Derivatives for the Targeted Therapy of Triple-Negative Breast Tumor Cells (MDA-MB-231) via EGFR/PI3K/AKT/mTOR Signaling Cascades
ArticleAbstract: Here, we described the synthesis of novel pyrazole-s-triazine derivatives via an easy one-pot procedPalabras claves:anticancer profile, apoptosis, DMF-DMA, EGFR/PI3K/AKT/mTOR, One-pot synthesis, pyrazolyl-s-triazineAutores:Al Zoubi M., Alberício F., Aldalbahi A., Alqudah D.A., Alshaer W., B. G. De la Torre, Barakat A., Daoud F., El-Faham A., Hatmal M.M., Haukka M., Nafie M.S., Sharma A., Shawish I.Fuentes:scopusAmide Formation: Choosing the Safer Carbodiimide in Combination with OxymaPure to Avoid HCN Release
ArticleAbstract: It has been reported that DIC can react with OxymaPure to render an oxadiazole compound with the conPalabras claves:Autores:Acosta G.A., Alberício F., B. G. De la Torre, El-Faham A., Luna O., Manne S.R., Orosz G., Royo M.Fuentes:scopusDesign and synthesis of mono-and di-pyrazolyl-s-triazine derivatives, their anticancer profile in human cancer cell lines, and in vivo toxicity in zebrafish embryos
ArticleAbstract: s-Triazine is considered a privileged structure, as it is found in several FDA-approved drugs. In thPalabras claves:anticancer activity, Pyrazole, S-triazine, Zebrafish embryosAutores:Al-Dhfyan A., Alberício F., Almarhoon Z.M., B. G. De la Torre, El-Faham A., Farooq M., Sharma A., Taha N.A., Wadaan M.A.M.Fuentes:scopusFormation of N <sup>α</sup>-terminal 2-dialkyl amino oxazoles from guanidinated derivatives under mild conditions
ArticleAbstract: Oxazole-containing peptides are an important class of molecules in medicinal chemistry programs. HerPalabras claves:Autores:Alberício F., B. G. De la Torre, El-Faham A., Kumar A., Mhlongo J.T., Monaim S.A.H.A.Fuentes:scopusGreen Solid-Phase Peptide Synthesis 2. 2-Methyltetrahydrofuran and Ethyl Acetate for Solid-Phase Peptide Synthesis under Green Conditions
ArticleAbstract: N,N-Dimethylformamide (DMF), N-methyl-2-pyrrolidone, and dichloromethane (DCM) are the most widely uPalabras claves:2-MeTHF, Green Chemistry, Peptide aggregation, Polyethylene glycol resins, Solid-phase peptide synthesis, solid-phase synthesisAutores:Acosta G.A., Alberício F., B. G. De la Torre, El-Faham A., Govender T., Jad Y.E., Kruger H.G.Fuentes:scopus