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2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis
ArticleAbstract: 2-MeTHF and CPME were evaluated as greener alternatives for the most employed solvents in peptide syPalabras claves:2-methyltetrahydrofuran, Cyclopentyl methyl ether, Green solvents, Peptide synthesis, Solid-phase peptide synthesisAutores:Acosta G.A., Alberício F., B. G. De la Torre, El-Faham A., Govender T., Jad Y.E., Khattab S.N., Kruger H.G.Fuentes:scopusDomino reactions with fluorinated five-membered heterocycles. α-Trifluoromethyl α-amino acids with unsaturated side-chains
ArticleAbstract: α-Trifluoromethyl α-amino acids with unsaturated side-chains have been prepared from 5-fluoro-4-trifPalabras claves:5-Fluoro-4-trifluoromethyloxazoles, Allyl alcohols, Claisen rearrangement, Farnesol, Geraniol, nucleophilic aromatic substitution, Propargyl alcohols, secondary structure, α-Trifluoromethyl α-amino acidsAutores:Alberício F., Burger K., Hennig L., Jan Spengler, Koksch B., Tsouker P.Fuentes:googlescopusNovel formulation of antimicrobial peptides enhances antimicrobial activity against methicillin-resistant Staphylococcus aureus (MRSA)
ArticleAbstract: Antimicrobial peptides (AMPs) have the ability to penetrate as well as transport cargo across bacterPalabras claves:Amps, Liposomes, MRSA, Peptide-lipidation, pH responseAutores:Agrawal N., Alberício F., B. G. De la Torre, Faya M., Govender T., Hazzah H.A., Maji R., Mocktar C., Nkambule B., Omolo C.A., Rambharose S., Walvekar P.Fuentes:scopusMicroreactors for peptide synthesis: Looking through the eyes of twenty first century!!!
OtherAbstract: The twenty first century has witnessed several advances in synthetic chemistry, among them microreacPalabras claves:Amide formation, Applications, Continuous flow, Microreactors, Peptide synthesisAutores:Alberício F., B. G. De la Torre, Cherkupally P., Govender T., Kruger H.G., Ramesh S.Fuentes:scopusSolid-phase peptide synthesis (SPPS), C-terminal vs. side-chain anchoring: A reality or a myth
OtherAbstract: Here we review the strategies for the solid-phase synthesis of peptides starting from the side chainPalabras claves:C-terminal acid peptide, Side-chain anchoring, Solid-phase peptide synthesis, Stepwise elongationAutores:Acosta G.A., Alberício F., B. G. De la Torre, Cherkupally P., Govender T., Kruger H.G., Ramesh S.Fuentes:scopusSynthesis of orthogonally protected l-threo-β-ethoxyasparagine
ArticleAbstract: Orthogonally protected l-threo-β-ethoxyasparagine (Fmoc-EtOAsn(Trt)- OH, 1) was synthesized from diePalabras claves:2,4,6-Trimethoxybenzylamide, amino acids, Hexafluoroacetone, peptide, TritylamideAutores:Alberício F., Jan Spengler, Pelay M., Tulla-Puche J.Fuentes:googlescopusSynthesis of α-trifluoromethyl α-amino acids with aromatic, heteroaromatic and ferrocenyl subunits in the side chain
ArticleAbstract: 5-Benzyloxy-4-trifluoromethyl-1,3-oxazoles, obtained from 5-fluoro-4-trifluoromethyloxazoles and benPalabras claves:1,3-Benzyl group migration versus Claisen rearrangement, 5-Fluoro-4-trifluoromethyl-1,3-oxazoles, Nucleophilic heteroaromatic substitution, Synthetic Tfm-Gly equivalent, α-Trifluoromethylamino acidsAutores:Alberício F., Burger K., Hennig L., Jan Spengler, Koksch B., Tsouker P.Fuentes:googlescopus