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Discovery of mitogen-activated protein kinase-interacting kinase 1 inhibitors by a comprehensive fragment-oriented virtual screening approach
ArticleAbstract: Mitogen-activated protein kinase-interacting kinases 1 and 2 (MNK1 and MNK2) phosphorylate the oncogPalabras claves:Autores:Albarran M.I., Antonio Salgado, Bischoff J.R., Corrionero A., Fominaya J., Mateos G., Oyarzabal J., Palacios I., Pastor J., Rabal O., Reymundo I., Urbano-Cuadrado M., Zarich N.Fuentes:scopusNew use of bis(benzotriazolyl)-1,2-(dialkylamino)ethanes for the synthesis of 2-H-3-dialkylamino imidazo[1,2-a]pyrazine derivatives
ArticleAbstract: First direct synthesis of 2-H-3-N-dialkyl-imidazo[1,2-a]pyrazines is described. This approach makesPalabras claves:2-H-3-N-Dialkyl-imidazo[1,2-a]pyrazines synthesis, Benzotriazole, One pot cyclisationAutores:Antonio Salgado, Hernández A.I., Martínez S.M., Pastor J., Rodríguez-Arístegui S., Varela C.Fuentes:scopus