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Novel substituted quinazolines for potent EGFR tyrosine kinase inhibitors
ArticleAbstract: The type I receptor tyrosine kinases (RTKs) are involved in various aspects of cell growth, survivalPalabras claves:Antitumour, Bioisostere, eGFR, Erlotinib, Gefitinib, HER-2, Quinazoline, Tyrosine kinase inhibitorAutores:Campos J.M., Conejo-García A., Cruz-López O., Fátima Morales, García-Rubino M.E., Gómez-Pérez V., Kimatrai M., Núnez M.C.Fuentes:scopusP-Nitrobenzenesulfonamides and their fluorescent dansylsulfonamides derived from N-alkylated o-(purine-methyl)anilines as novel antitumour agents
ArticleAbstract: We have designed and synthesized a novel series of fourteen alkylated purines with notable in vitroPalabras claves:Autores:Campos J.M., Conejo-García A., Fátima Morales, Marchal J.A., Morata C., Ramírez A.Fuentes:scopus