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scopus(23)
Characterization of the activation pathway of phosphoramidate triester prodrugs of stavudine and zidovudine
ArticleAbstract: The phosphoramidate triester prodrugs of anti-human HIV 2',3'- dideoxynucleoside analogs (ddN) reprePalabras claves:Autores:Antonio Salgado, Balzarini J., Cahard D., De Clercq E., McGuigan C., Naesens L., Pathirana R., Saboulard D., Velázquez S.Fuentes:scopusComplexation of daclatasvir by single isomer methylated β-cyclodextrins studied by capillary electrophoresis, NMR spectroscopy and mass spectrometry
ArticleAbstract: In capillary electrophoresis an enantioseparation of daclatasvir (DCV) was observed in case of heptaPalabras claves:capillary electrophoresis, Complex stoichiometry, Complex structure, Cyclodextrin-analyte complexation, Mass spectrometry, nuclear magnetic resonance spectroscopyAutores:Antonio Salgado, Benkovics G., Chankvetadze B., Krait S., Malanga M., Naumann L., Neusüß C., Peluso P., Scriba G.K.E., Sohajda T.Fuentes:scopusBi- and bisbibenzyls from the roots of Dichapetalum heudelotii and their antiproliferative activities
ArticleAbstract: Two new bisbibenzyls, heudelotol A (1) and B (2), along with the known bibenzyls, (E)-combretastatinPalabras claves:antiproliferative activity, Bisbibenzyls, Combretastatins, Dichapetalaceae, Dichapetalum heudelotiiAutores:Antonio Salgado, Chama M.A., Dziwornu G.A., Osei-Safo D., Sunassee S.N.Fuentes:scopusA cascade reaction of azolopyrimidines. Synthesis of unusual indole and azaindole derivatives
ArticleAbstract: The reaction of bromo substituted pyrido[3−,2−:4,5]pyrrolo-[1,2-c]pyrimidine and pyrimido[1,6-a]indoPalabras claves:Autores:Alvarez-Builla J., Antonio Salgado, Burgos C., Morón M., Mosquer M.E.G., Vaquero J.J.Fuentes:scopusFormation, Characterization, and Occurrence of β-Carboline Alkaloids Derived from α-Dicarbonyl Compounds and l -Tryptophan
ArticleAbstract: β-Carbolines (βCs) are naturally occurring bioactive alkaloids, whereas α-dicarbonyl compounds are rPalabras claves:3-deoxyglucosone, advanced glycation, glyoxal, Maillard reaction, methylglyoxal, tryptophan, α-dicarbonyl-derived βCs, α-dicarbonyls, β-carboline alkaloidsAutores:Antonio Salgado, Herraiz M., Herraiz T., Mateo H., Peña A.Fuentes:scopusFragment-Hopping-Based Discovery of a Novel Chemical Series of Proto-Oncogene PIM-1 Kinase Inhibitors
ArticleAbstract: A new chemical series, triazolo[4,5-b]pyridines, has been identified as an inhibitor of PIM-1 by a cPalabras claves:Autores:Albarran M.I., Alvarez R.M., Antonio Salgado, Bischoff J.R., Blanco C., Kurz G., Ortega M.A., Oyarzabal J., Pastor J., Pevarello P., Rabal O., Saluste G.Fuentes:scopusElectrosynthesis of Oxazol-2(3H)-Ones and Diaroylhydrazines from 1,2-Dicarbonyl Compounds and Arenediazonium Salts
ArticleAbstract: New five-membered oxazol-2(3H)-one heterocycles and 1,2-diaroylhydrazines are obtained in good yieldPalabras claves:1,2-diaroylhydrazines, 3-methyl-oxazol-2(3H)-ones, electrochemical reduction, N-methylformamide, radical couplingAutores:Antonio Salgado, Barba F., Batanero B., Quirós I.Fuentes:scopusEnantiomeric separation of the antiuremic drug colchicine by electrokinetic chromatography. Method development and quantitative analysis
ArticleAbstract: Two analytical methodologies were developed by CE enabling the enantiomeric separation of colchicinePalabras claves:capillary electrophoresis, colchicine, enantiomer migration order, Enantioseparation, H NMR, QuantitationAutores:Antonio Salgado, Castro-Puyana M., García M.Á., Marina M.L., Menéndez-López N., Valimaña-Traverso J.Fuentes:scopusNew use of bis(benzotriazolyl)-1,2-(dialkylamino)ethanes for the synthesis of 2-H-3-dialkylamino imidazo[1,2-a]pyrazine derivatives
ArticleAbstract: First direct synthesis of 2-H-3-N-dialkyl-imidazo[1,2-a]pyrazines is described. This approach makesPalabras claves:2-H-3-N-Dialkyl-imidazo[1,2-a]pyrazines synthesis, Benzotriazole, One pot cyclisationAutores:Antonio Salgado, Hernández A.I., Martínez S.M., Pastor J., Rodríguez-Arístegui S., Varela C.Fuentes:scopusNovel biologically active dihydroxycinnamate-derived polyether from different species of family Boraginaceae
ArticleAbstract: Plants belonging to Boraginaceae family such as Symphytum asperum, S.caucasicum, S.officinale and AnPalabras claves:Anchusa, Boraginaceae, Dihydroxycinnamate-derived polyether, NMR, Poly[3-(3,4-dihydroxyphenyl)glyceric acid], poly[oxy-1-carboxy-2-(3,4-dihydroxyphenyl)ethylene], SymphytumAutores:Amiranashvili L., Antonio Salgado, Barbakadze V., Chankvetadze B., Gogilashvili L., Merlani M., Mulkijanyan K.Fuentes:scopus