Documentos de B. G. De la Torre | REDI

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Filtros aplicados

Publisher: "Tetrahedron Letters"

Subtipo de publicación

Área temáticas

Química orgánica(5)

Química física(4)

Farmacología y terapéutica(3)

Química analítica(3)

Área de conocimiento

Ingeniería química(5)

Ciencia de materiales(2)

Síntesis química(2)

Año de Publicación

Origen

Palabras Claves

Solid-phase peptide synthesis(6)

cyclic peptides(2)

Antimicrobial peptide(1)

Bzl protecting group(1)

Carbodiimides(1)

An improved and efficient strategy for the total synthesis of a colistin-like peptide

Abstract: Polymyxins have re-emerged as the last-line therapy for treatment against extremely multi-drug resis

Palabras claves:

Antimicrobial peptide, colistin, Convergent method, Synthesis

Alberício F., B. G. De la Torre, Govender T., Kruger H.G., Ramesh S.

Green solid-phase peptide synthesis 4. γ-Valerolactone and N-formylmorpholine as green solvents for solid phase peptide synthesis

Abstract: Herein, we report the use of γ-valerolactone (GVL) and N-formylmorpholine (NFM) as DMF substitutes i

Palabras claves:

Green solvents, GVL, NFM, polystyrene resin, Solid-phase peptide synthesis

Alberício F., B. G. De la Torre, El-Faham A., Jad Y.E., Kumar A.

Facile solid-phase synthesis of head-side chain cyclothiodepsipeptides through a cyclative cleavage from MeDbz-resin

Abstract: Head to side-chain cyclothiodepsipeptides were conveniently prepared through a cyclative cleavage us

Palabras claves:

cyclic peptides, On resin cyclization, Solid-phase peptide synthesis, Thiolactone, Thiopeptides

Acosta G.A., Alberício F., B. G. De la Torre, Royo M.

Oxyma-T, expanding the arsenal of coupling reagents

Abstract: Herein, we report a new oxime-based additive (Oxyma-T) with a similar structure to HONM and Oxyma-B

Palabras claves:

Carbodiimides/additives, Oxime, Peptide coupling reagent, Solid-phase peptide synthesis, Solution-phase peptide synthesis

Alberício F., B. G. De la Torre, El-Faham A., Govender T., Jad Y.E., Kruger H.G.

Incorporation of pseudoproline monomer (Fmoc-Thr[ψ<sup>Me,Me</sup>pro]–OH) facilitates efficient solid-phase synthesis of difficult peptides

Abstract: Solid-Phase Peptide Synthesis (SPPS) is a convenient and efficient method by which to prepare peptid

Palabras claves:

Chain to chain interaction, Deletion peptides, hGH peptide, JR Peptide, SPPS

Alberício F., B. G. De la Torre, Bruckdorfer T., Manne S.R., Rustler K.

Minimizing side reactions during amide formation using DIC and oxymapure in solid-phase peptide synthesis

Abstract: N,N’-diisopropylcarbodiimide (DIC) and OxymaPure are the reagents of choice for the formation of pep

Palabras claves:

Carbodiimides, HCN formation, Oxadiazole, Side-reaction, Solid-phase peptide synthesis

Alberício F., B. G. De la Torre, El-Faham A., Manne S.R.

γ-Valerolactone (GVL): An eco-friendly anchoring solvent for solid-phase peptide synthesis

Abstract: Due to the hazardous nature of CH2Cl2, regulatory authorities have imposed restrictions to minimize

Palabras claves:

Dipeptide formation, Green Chemistry, Racemization, Wang resin

Al Musaimi O., Alberício F., B. G. De la Torre, Basso A., El-Faham A.

Solid-phase N-glycopeptide synthesis using allyl side-chain protected Fmoc-amino acids

Abstract: A method for the preparation of glycopeptides using a three-dimensional orthogonal solid-phase strat

Palabras claves:

allyl esters, glycopeptides, Orthogonal protection, solid-phase synthesis

Alberício F., B. G. De la Torre, Eritja R., Kates S.

Solid-phase synthesis of homodetic cyclic peptides from Fmoc-MeDbz-resin

Abstract: Cyclic homodetic peptides are very appealing for medicinal chemistry programs. In addition to the hi

Palabras claves:

Cyclactive cleavage, cyclic peptides, MeDbz linker, Solid-phase peptide synthesis

Acosta G.A., Alberício F., B. G. De la Torre, El-Faham A., Monaim S.A.H.A., Royo M.

Solid-phase synthesis of peptides containing 1-Hydroxypyridine-2-one (1,2-HOPO)

Abstract: Herein a friendly method for the preparation of 1-hydroxypyridine-2-one (1,2-HOPO)-containing peptid

Palabras claves:

Bzl protecting group, Fe(III) chelating compounds, Siderophores, Solid-phase peptide synthesis, Trifluoromethanesulfonic acid

Al Shaer D.M., Alberício F., B. G. De la Torre