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Alkyl-linked bis-THTT derivatives as potent in vitro trypanocidal agents
ArticleAbstract: The effect of several alkyl-linked bis tetrahydro-(2H)-1,3,5-thiadiazine-2- thione (bis-THTT) on LeiPalabras claves:Alkyl-linked bis-THTT anti-protozoal activityAutores:Alvarez A., Atherton R., Coro J., Hortensia Rodriguez Cabrera, Little S., Perez-Pineiro R., Suárez Navarro M., Wharton H., Yardley V.Fuentes:googlescopusIn vitro activities of thiadiazine derivatives against Leishmania amazonensis
ArticleAbstract: Ten thiadiazine derivatives were tested in vitro for antiparasitic effects against both extracellulaPalabras claves:Antiparasitic drugs, Leishmania amazonensis, amastigotes, promastigotes, Thiadiazine derivatives, antileishmanial activity in vitro, toxicityAutores:Fonseca L., Hortensia Rodriguez Cabrera, Montalvo Álvarez A.M., Monzote L., Perez-Pineiro R., Suárez Navarro M.Fuentes:googlescopusIn vitro and in vivo assays of 3,5-disubstituted-tetrahydro-2H-1,3,5-thiadiazin-2-thione derivatives against Trypanosoma cruzi
ArticleAbstract: Cytotoxicity assays of 24 new 3,5-disubstituted-tetrahydro-2H-1,3,5-thiadiazin-2-thione derivativesPalabras claves:AMASTIGOTES, Antichagasic drugs, Antitrypanosomal activity assays, Cytotoxicity assays, J774 macrophages, Thiadiazine thione derivativesAutores:García-Trevijano J.A.E., Gómez-Barrio A., Hortensia Rodriguez Cabrera, Muelas S., Ochoa C., Perez-Pineiro R., Suárez Navarro M.Fuentes:googlescopusSynthesis and antiprotozoal evaluation of new N<sup>4</sup>-(benzyl) spermidyl-linked bis(1,3,5-thiadiazinane-2-thiones)
ArticleAbstract: The synthesis and in-vitro antiprotozoal evaluation of novel N 4-(benzyl)spermidyl-linked bis(1,3,5-Palabras claves:1,3,5-thiadiazinane-2-thione, Protozoocidal activity, SpermidineAutores:Coro J., Hortensia Rodriguez Cabrera, Little S., Martín N., Perez-Pineiro R., Súrez M., Yardley V.Fuentes:scopusSynthesis and antiprotozoan evaluation of new alkyl-linked bis(2-thioxo-[1,3,5]thiadiazinan-3-yl) carboxylic acids
ArticleAbstract: Two new series of several alkyl-linked bis(2-thioxo-[1,3,5]thiadiazinan-3- yl) carboxylic acids werePalabras claves:Antiparasitics, chemotherapy, Thiadiazine-2-thioneAutores:Coro J., Gómez-Barrio A., Hortensia Rodriguez Cabrera, Montero D., Nogal-Ruiz J.J., Perez-Pineiro R., Rolón M.S., Suárez Navarro M., Vega C.Fuentes:scopus