Documentos de Kumar A. | REDI

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Área temáticas: "Química orgánica"

Subtipo de publicación

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Organic Process Research and Development(2)

Bioorganic Chemistry(1)

Área temáticas

Farmacología y terapéutica(5)

Química física(4)

Tecnología de productos químicos industriales(3)

Ingeniería química(2)

Química y ciencias afines(2)

Área de conocimiento

Química orgánica(5)

Ingeniería química(4)

Síntesis química(2)

Año de Publicación

Origen

Palabras Claves

Solid-phase peptide synthesis(4)

Green solvent(3)

4-methylpiperidine(1)

Acyl piperidide(1)

1,3,5-Triazine as core for the preparation of dendrons

Abstract: A unique property of 2,4,6-trichloro-1,3,5-triazine (TCT) is its ability to undergoes a nucleophilic

Palabras claves:

1+2 mode, Dendron, HPLC, Nucleophiles, S-triazine

Alberício F., B. G. De la Torre, El-Faham A., Kumar A., Sharma A., Sheyi R.

Diethylphosphoryl-oxymab (DEPO-B) as a solid coupling reagent for amide bond formation

Abstract: A new phosphonium based coupling reagent DEPO-B has been synthesized from 5-(hydroxyimino)-1,3-dimet

Palabras claves:

coupling reagent, Diethylphosphoryl-OxymaB, Hydrolytic stability, Phosphonium salts, SOLUBILITY

Alberício F., B. G. De la Torre, El-Faham A., Jad Y.E., Kumar A.

Formation of N <sup>α</sup>-terminal 2-dialkyl amino oxazoles from guanidinated derivatives under mild conditions

Abstract: Oxazole-containing peptides are an important class of molecules in medicinal chemistry programs. Her

Palabras claves:

Alberício F., B. G. De la Torre, El-Faham A., Kumar A., Mhlongo J.T., Monaim S.A.H.A.

Exploiting azido-dichloro-triazine as a linker for regioselective incorporation of peptides through their N, O, S functional groups

Abstract: In the field of bioconjugation, linker development has witnessed massive growth in recent years. 2,4

Palabras claves:

Bioconjuation, Linker, Orthogonal chemoselectivity, Orthogonality, Solid-phase peptide synthesis

Alberício F., B. G. De la Torre, El-Faham A., Kumar A., Sharma A.

Fmoc-Amox, A Suitable Reagent for the Introduction of Fmoc

Abstract: Synthesis of most peptides is achieved using solid-phase peptide synthesis employing the Fmoc/tert-b

Palabras claves:

Alberício F., B. G. De la Torre, El-Faham A., Haimov E., Kumar A., Sharma A.

N-Butylpyrrolidinone for Solid-Phase Peptide Synthesis is Environmentally Friendlier and Synthetically Better than DMF

Abstract: Solid-phase peptide synthesis (SPPS) is the method of choice for the preparation of peptides in both

Palabras claves:

aspartimide formation, Green solvent, N-butylpyrrolidinone, Racemization, Solid-phase peptide synthesis

Alberício F., Alhassan M., B. G. De la Torre, Kumar A., Lopez J.

N-methylation in amino acids and peptides: Scope and limitations

Abstract: Active pharmaceutical ingbkp_redients (APIs) can be divided into two types, namely chemical and biol

Palabras claves:

cyclic peptides, NMAA, side-reactions, Solid-phase peptide synthesis

Alberício F., B. G. De la Torre, El-Faham A., Jad Y.E., Kumar A., Monaim S.A.H.A., Sharma A.

Liquid-Phase Peptide Synthesis (LPPS): A Third Wave for the Preparation of Peptides

Abstract: Since the last century, peptides have gained wide acceptance as drugs, with almost 100 already in th

Palabras claves:

Alberício F., B. G. De la Torre, Kumar A., Sharma A.

Investigating Triorthogonal Chemoselectivity. Effect of Azide Substitution on the Triazine Core

Abstract: An example of triorthogonal chemoselectivity is reported here for the first time. In this regard, a

Palabras claves:

Alberício F., B. G. De la Torre, El-Faham A., Kumar A., Sharma A., Sheyi R.

Jetting manufacturing of resins for solid-phase peptide synthesis

Abstract: Peptides are an important class of Active Pharmaceutical Ingbkp_redients. Indeed, it is now feasible

Palabras claves:

loading, peptide synthesis., Resins, SPPS, styrene/DVB, swelling

Alberício F., B. G. De la Torre, Basso A., Jad Y.E., Ji C., Kumar A., Ma Z., Musaimi O.A.L., Serban S.