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scopus(11)
Barbiturate- And Thiobarbituarte-Based s-Triazine Hydrazone Derivatives with Promising Antiproliferative Activities
ArticleAbstract: A new class of compounds, which include s-triazine with pyrimidinetrione or thiopyrimidinedione moiePalabras claves:Autores:Al-Rasheed H.H., Alberício F., B. G. De la Torre, Dahlous K.A., El-Faham A., Sharma A., Sholkamy E.N.Fuentes:scopus1,3,5-Triazino Peptide Derivatives: Synthesis, Characterization, and Preliminary Antileishmanial Activity
ArticleAbstract: A library of short di-, tri-, and tetra-peptides with an s-triazine moiety at the N terminus and eitPalabras claves:1,3,5-triazine derivatives, antileishmanial compounds, morpholines, Peptides, piperidinesAutores:Abd El-Rahman M.M., Alberício F., B. G. De la Torre, Bekhit A.A., El-Faham A., Khalil H.H., Khattab S.N.Fuentes:scopusCorrigendum: Pyrazolyl-s-triazine with indole motif as a novel of epidermal growth factor receptor/cyclin-dependent kinase 2 dual inhibitors(Front. Chem., (2022), 10, (1078163), 10.3389/fchem.2022.1078163)
OtherAbstract: In the original article, there was an error in the Affiliation for Samha Al Ayoubi2. Instead of “SamPalabras claves:anticancer profile, apoptosis, EGFR/CDK-2, ÍNDOLE, pyrazolyl-s-triazineAutores:Al Ayoubi S., Al Zoubi M., Al-Rasheed H.H., Alberício F., Aldalbahi A., Ali M., Alshaer W., B. G. De la Torre, Barakat A., El-Faham A., Nafie M.S., Shawish I.Fuentes:scopusAcetic Acid Mediated for One-Pot Synthesis of Novel Pyrazolyl s-Triazine Derivatives for the Targeted Therapy of Triple-Negative Breast Tumor Cells (MDA-MB-231) via EGFR/PI3K/AKT/mTOR Signaling Cascades
ArticleAbstract: Here, we described the synthesis of novel pyrazole-s-triazine derivatives via an easy one-pot procedPalabras claves:anticancer profile, apoptosis, DMF-DMA, EGFR/PI3K/AKT/mTOR, One-pot synthesis, pyrazolyl-s-triazineAutores:Al Zoubi M., Alberício F., Aldalbahi A., Alqudah D.A., Alshaer W., B. G. De la Torre, Barakat A., Daoud F., El-Faham A., Hatmal M.M., Haukka M., Nafie M.S., Sharma A., Shawish I.Fuentes:scopusExploiting the Thiobarbituric Acid Scaffold for Antibacterial Activity
ArticleAbstract: Thiobarbituric acid (TBA) has been considered a privileged structure for developing antimicrobial agPalabras claves:Antibiotics, barbituric acid, nanoformulations, Thiobarbituric acidAutores:Alberício F., Almarhoon Z.M., B. G. De la Torre, El-Faham A., Hazzah H.A., Noki S., Sharma A., Zamisa S.J.Fuentes:scopusEnamine barbiturates and thiobarbiturates as a new class of bacterial urease inhibitors
ArticleAbstract: Urease is a therapeutic target associated with several important diseases and health problems. BasedPalabras claves:Barbituric, DFT, Pyrimidine-trione, Thiobarbituric, Urease inhibitorsAutores:Al-Majid A.M., Alberício F., Ali M., Ashraf S., B. G. De la Torre, Barakat A., Choudhary M.I., El-Faham A., Ul-Haq Z., Yousuf S.Fuentes:scopusNovel 4,6-disubstituted s-triazin-2-yl amino acid derivatives as promising antifungal agents
ArticleAbstract: A novel series of 4,6-disubstituted s-triazin-2-yl amino acid derivatives was prepared and characterPalabras claves:2,4,6-trichlorotriazine, Antifungal, Candida Albicans, N-myristoltransferase, TCT, Triazine amino acidAutores:Alberício F., Alhameed R.A., Almarhoon Z.M., B. G. De la Torre, El-Faham A., Khan S.A., Sharma A., Sholkamy E.N., Ul-Haq Z.Fuentes:scopusS-triazine: A privileged structure for drug discovery and bioconjugation
ArticleAbstract: This review provides an overview of the broad applicability of s-triazine. Our many years working wiPalabras claves:azide, Nucleophiles, Orthogonal chemoselectivity, S-triazineAutores:Alberício F., B. G. De la Torre, El-Faham A., Sharma A., Sheyi R.Fuentes:scopusSynthesis and Antiproliferative Activity of a New Series of Mono- A nd Bis(dimethylpyrazolyl)-s-triazine Derivatives Targeting EGFR/PI3K/AKT/mTOR Signaling Cascades
ArticleAbstract: Here, we synthesized a newseries of mono- A nd bis(dimethylpyrazolyl)-s-triazine derivatives. The syPalabras claves:Autores:Alberício F., Albohy A., Aldalbahi A., B. G. De la Torre, Barakat A., Bekhit A.A., El-Faham A., Haukka M., Khan A., Malebari A.M., Nafie M.S., Shawish I., Ul-Haq Z.Fuentes:scopusSynthesis and Biological Evaluation of a Teixobactin Analogue
ArticleAbstract: The first synthesis and biological activity of a teixobactin analogue is reported. Substitution of tPalabras claves:Autores:Acosta G.A., Alberício F., B. G. De la Torre, El-Faham A., Govender T., Jad Y.E., Kruger H.G., Naicker T., Ramtahal M.Fuentes:scopus